Discuss This Drug

paliperidone

CHEBI:CHEBI_82978

Definition

A racemate comprising equimolar amounts of (R)- and (S)-paliperidone. Paliperidone is the primary active metabolite of the older antipsychotic risperidone and is used for treatment of schizophrenia.

Chemical Information

Molecular Formula
C23H27FN4O3
Molecular Mass
426.48390
Charge
0

Alternative Names

  • (+-)-paliperidone
  • (RS)-paliperidone
  • 9-hydroxy-risperidone
  • 9-Hydroxyrisperidone
  • 9-OH-risperidone
  • Invega
  • paliperidone
  • R 76477
  • R-76477
  • rac-3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-9-hydroxy-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one
  • rac-paliperidone
  • racemic paliperidone
  • Ro-76477
  • RO76477

Treatment Applications

Drug Classification

Important Medical Information

⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.

  • Always consult with a healthcare professional before starting, stopping, or modifying any medication.
  • Side effects may vary and this list may not be comprehensive.
  • Drug interactions may occur with other medications.

Additional Identifiers

DRON_00010000
679314
oboInOwl#hasDbXref
Wikipedia:Paliperidone
core#notation
CHEBI:82978

Additional References

Wikipedia:Paliperidone

🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.

Additional Attributes

product_type
BULK INGREDIENT
marketing_category
BULK INGREDIENT FOR HUMAN PRESCRIPTION COMPOUNDING
dosage_form
INJECTION, SUSPENSION, EXTENDED RELEASE
labeler_name
Sintenovo SA de CV
application_number
ANDA208643
product_ndc
42291-916
oboInOwl#hasOBONamespace
chebi_ontology
DRON_00010000
679314
oboInOwl#hasDbXref
Wikipedia:Paliperidone
oboInOwl#id
CHEBI:82978
generic_name
PALIPERIDONE PALMITATE (STERILE)
brand_name
INVEGA HAFYERA
brand_name_base
INVEGA HAFYERA
RO_0000087
http://purl.obolibrary.org/obo/CHEBI_37955
oboInOwl#inSubset
http://purl.obolibrary.org/obo/chebi#3_STAR
BFO_0000051
http://purl.obolibrary.org/obo/CHEBI_83806
rxcui
2570421
package_marketing_start_date
20-AUG-13
manufacturer_name
Camber Pharmaceuticals, Inc
package_description
30 TABLET, EXTENDED RELEASE in 1 BOTTLE (16714-866-01)
active_ingredient_strength
546 mg/1.75mL
nui
N0000175430
pharm_class_epc
Atypical Antipsychotic [EPC]
active_ingredient_name
PALIPERIDONE PALMITATE
unii
R8P8USM8FR
spl_set_id
6cd61892-d2cb-434d-83ed-5c1b2c4e7a0b
upc
0368180526063
package_ndc
50458-550-01
listing_expiration_date
20241231
route
INTRAMUSCULAR
marketing_start_date
20111205
spl_id
1f346295-d7db-6347-4606-f24dfc78397c
core#notation
CHEBI:82978
pharm_class
Atypical Antipsychotic [EPC]
22-rdf-syntax-ns#type
http://www.w3.org/2002/07/owl#Class
rdf-schema#range
https://w3id.org/def/predibionto#has_drug_113845
has_treatment
http://purl.obolibrary.org/obo/DOID_13969
rdf-schema#domain
https://w3id.org/def/predibionto#has_side_effect36518
owl#annotatedSource
t307596
owl#someValuesFrom
t2884797